Synthesis and Biological Evaluation of N-Heterocyclic Substituted Fluoro-Benzothiazole Sulphonamido Analogs as a Potential Therapeutic Agents
نویسندگان
چکیده
The present investigation is aimed to synthesize fluorobenzothiazole comprising sulphonamido pyrazole analogs starting from fluoro-chloroaniline get 2-amino-6-fluoro-7-chloro (1,3) benzothiazole (I), this was treated with anilino-s-methyl ethylene cyanoacetamide in the presence of ethanol desired molecules. synthesized targeted molecules are characterized, docked and screened for their invitro antidiabetic properties.
 Keywords: Fluorobenzothiazole, Docking,
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ژورنال
عنوان ژورنال: Journal of Biomedical and Pharmaceutical Research
سال: 2022
ISSN: ['2279-0594', '2589-8752']
DOI: https://doi.org/10.32553/jbpr.v11i1.893